找到约 30 条 “Calcium Channel” 相关结果 (用时 0.085 秒)
目录号 | 产品名称 | 中文名称 | 靶点 |
---|---|---|---|
M2248 | Cilnidipine | 西尼地平 | Calcium Channel |
FRC 8653 | |||
Cilnidipine是一种钙离子通道(Calcium Channel)抑制剂。 | |||
M2820 | Lomerizine dihydrochloride | 盐酸洛美利嗪 | Calcium Channel |
KB-2796 | |||
Lomerizine 2HCl是一种相对新型L-和T-型钙通道(Calcium Channel)阻滞剂。 | |||
M3118 | Verapamil hydrochloride | 盐酸维拉帕米 | Calcium Channel |
(±)-Verapamil hydrochlorid | |||
Verapamil hydrochloride是一种具有口服活性的L-型钙通道(Calcium Channel)抑制剂,可以消除钙通道激动剂诱导的钙内流和细胞凋亡。Verapamil hydrochloride 也是一种有效的口服活性的第一代 P 糖蛋白 (P-gp) 抑制剂。维拉帕米能抑制 CAT1 介导的精氨酸、高精氨酸和 ADMA 的吸收,其 IC50 值分别为 85.3、58.1 和 113 µM。 | |||
M3296 | Manidipine dihydrochloride | 盐酸马尼地平 | Calcium Channel |
CV-4093 | |||
Manidipine 2HCl是Manidipine的盐酸盐形式,是钙通道(Calcium Channel)阻断剂,IC50为2.6 nM。 | |||
M3498 | Nimodipine | 尼莫地平 | Calcium Channel |
BAY-e 9736 | |||
Nimodipine是一种二氢吡啶衍生物,是钙离子通道抑制剂(Calcium Channel)Nifedipine的类似物,具有降压活性。Nimodipine能减少细胞内游离Ca2+,Beclin-1及细胞自噬。 | |||
M3500 | Diltiazem hydrochloride | 地尔硫;硫氮卓酮;恬尔心;盐酸地尔硫卓 | Calcium Channel |
CRD-401 | |||
Diltiazem hydrochloride(地尔硫,硫氮卓酮,恬尔心,酸地尔硫卓)是一种钙通道(Calcium Channel)阻滞剂,对细胞外钙离子的跨膜流入具有抑制作用,可用于肿瘤及心血管疾病的相关研究。 | |||
M3613 | NP118809 | NP118809 | Calcium Channel |
39-1B4, NP-118809 | |||
NP-118809 (39-1B4)是一种有效的n型钙通道(Calcium Channel)阻滞剂(IC50= 0.11 uM);l型钙通道具有良好的选择性。 | |||
M3959 | Felodipine | 非洛地平 | Calcium Channel |
CGH-869 | |||
Felodipine是一种l型Ca2+通道(Calcium Channel)阻滞剂,比N-、R-、P/Q-和t型通道有选择性,IC50为0.15 nM。此外,Felodipine还能通过抑制细胞Ca2+摄取,导致钙蛋白酶活性降低,从而水解Atg5,成为细胞自噬的负调控因子。可用于原发性高血压的相关研究。 | |||
M4968 | Mitiglinide calcium hydrate | 米格列奈钙 | Potassium Channel |
KAD-1229 calcium hydrate; S-21403 calcium hydrate | |||
Mitiglinide calcium hydrate is a drug for the treatment of type 2 diabetes; it is a highly selective KATP channel antagonist. | |||
M5073 | (R)-(+)-BAY K 8644 | (R)-(+)-BAY K 8644 | Calcium Channel |
(R)-(+)-Bay-K-8644; R-4407; NI-105; (+)-BAY-K-8644; Bayk8644 | |||
(R)-(+)-BAY K 8644 是一种钙通道(calcium channel)抑制剂,抑制 Ba2+电流 (IBa) ,IC50为975 nM。同时,(R)-(+)-BAY K 8644也是一种有效的TMEM176B抑制剂。此外,(R)-(+)-BAY K 8644还能提高Oct4和Klf4对小鼠成纤维细胞的重编程效率,弥补Sox2缺失带来的影响。 | |||
M5080 | Efonidipine hydrochloride | 依福地平盐酸盐 | Calcium Channel |
NZ-105 | |||
Efonidipine Hcl is a dual T-type and L-type calcium channel blocker . | |||
M5139 | Amlodipine | 氨氯地平 | Calcium Channel |
UK-48340 | |||
Amlodipine 是一种具有口服活性的二氢吡啶钙通道(Calcium Channel)阻滞剂,通过阻断电压依赖性的 L 型钙通道,从而抑制钙离子内流。 | |||
M5756 | L-Phenylalanine | L-Phenylalanine | Calcium Channel |
(S)-2-Amino-3-phenylpropionic acid | |||
L-Phenylalanine (L-苯丙氨酸)是α2δ钙离子通道(Calcium Channel)拮抗剂,Ki为980 nM。 | |||
M6499 | Bepridil hydrochloride | 盐酸贝普地尔 | Calcium Channel |
CERM 1978 | |||
Bepridil hydrochloride (CERM 1978) 是一种钙离子通道 (calcium channel) 抑制剂,可以用于心绞痛的研究。 | |||
M7723 | CBIQ | CBIQ | Others |
CBIQ is an activator of the cystic fibrosis transmembrane conductance regulator (CFTR) and the intermediate-conductance calcium-sensitive K+ channel (KCNN4). | |||
M7898 | Lidoflazine | 利多氟嗪 | Others |
Lidoflazine is an antianginal calcium channel blocker that carries a significant risk of QT interval prolongation and ventricular arrhythmia. | |||
M7906 | MRS 1845 | MRS 1845 | Others |
Store-operated calcium (SOC) channel inhibitor. | |||
M8315 | Ralfinamide mesylate | Ralfinamide mesylate | Others |
Ralfinamide is a mixed sodium and N-type calcium channel blocker. | |||
M8330 | Carboxyamidotriazole | Carboxyamidotriazole | Others |
Carboxyamidotriazole (L-651582) is an orally active calcium channel blocker. | |||
M8515 | Nifetepimine | Nifetepimine | Others |
Nifetepimine is a dihydropyrimidone calcium channel blocker that down-modulates SERCA3 (sarco/endoplasmic reticulum Ca2+ -ATPase 3) pump, and protects of the CD4+ T cells from tumor-induced apoptosis. | |||
M14189 | Amlodipine maleate | 马来酸氨氯地平 | Calcium Channel |
Amlodipine maleate 是二氢吡啶类钙通道 (calcium channel) 阻滞剂,作为一种具有口服活性的抗心绞痛试剂 (antianginal agent)。Amlodipine maleate 阻断了电压依赖性的 L 型钙通道,从而抑制了钙离子内流。Amlodipine maleate 可用于高血压和癌症的研究。 | |||
M14201 | Mibefradil dihydrochloride | 盐酸米贝地尔 | Calcium Channel |
Ro 40-5967 dihydrochloride | |||
Mibefradil dihydrochloride (Ro 40-5967 dihydrochloride) 是一种钙离子通道 (calcium channel) 抑制剂,选择性作用于 T 型 Ca2+通道,作用于 T 型和 L 型通道,IC50 分别为 2.7 μM 和 18.6 μM。 | |||
M14203 | Norverapamil hydrochloride | 盐酸去甲维拉帕米 | Calcium Channel |
(±)-Norverapamil hydrochloride; D591 hydrochloride | |||
Norverapamil hydrochloride,是 Verapamil 的 N-去甲基代谢物,是一种钙通道 (L-type calcium channel) 阻滞剂和 P-糖蛋白 (P-gp) 功能抑制剂。 | |||
M14204 | Verapamil | 维拉帕米 | Calcium Channel |
(±)-Verapamil; CP-16533-1 | |||
Verapamil ((±)-Verapamil) 是一种钙通道 (calcium channel) 阻滞剂,是一种有效的口服活性的第一代 P 糖蛋白 (P-gp) 抑制剂。Verapamil 能也抑制 CYP3A4,并可用于高血压,心律不齐和心绞痛的研究。 | |||
M14514 | N-(p-amylcinnamoyl) Anthranilic Acid | N-(p-amylcinnamoyl) Anthranilic Acid | Phospholipase |
ACA | |||
N-(p-amylcinnamoyl) Anthranilic Acid (ACA) 是一种广谱磷脂酶 A2 (PLA2) 的抑制剂,TRP channel的阻滞剂。N-(p-amylcinnamoyl) Anthranilic Acid (ACA) 也是一种有效的钙离子激活氯通道 (calcium-activated chloride channels) 的可逆抑制剂,有潜力用于心律失常的相关研究。 | |||
M16986 | Kobusin | 去甲槟郎碱 | GLUT |
Kobusin(去甲槟郎碱)是从 Pnonobio biondii Pamp 分离的双环氧木脂素,同时也是 CFTR 和 CaCCgie 氯化物通道的激活剂,以及ANO1/CaCC (calcium-activated chloride channel) 通道的抑制剂。 | |||
M18297 | 14-Deoxyandrographolide | 14-去氧穿心莲内酯 | Calcium Channel |
14-Deoxyandrographolide 是一种具有钙通道 (calcium channel) 阻断活性的劳丹脂二萜。 | |||
M20409 | Levamlodipine | Levamlodipine | Calcium Channel |
S-amlodipine | |||
Levamlodipine is a pharmacologically active enantiomer of amlodipine which belongs to the dihydropyridine group of calcium channel blocker. It acts on the L-type of calcium channels and its treatment results in vasodilation and a fall in blood pressure. | |||
M20441 | Efonidipine | Efonidipine | Calcium Channel |
NZ-105 | |||
Efonidipine is an L- and T-type calcium channel blocker leading to vasodilation and decreased automaticity of the heart. It also suppresses aldosterone secretion from the adrenal. | |||
M20469 | Nicardipine | Nicardipine | Others |
YC-93 | |||
Nicardipine(YC-93) is a calcium channel blocker that has been widely used to control blood pressure in severe hypertension following events such as ischemic stroke, traumatic brain injury, and intracerebral hemorrhage. |
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